1: (3-bromopyridin-4-yl)-dimethyl-amine With isopropylmagnesium chloride in tetrahydrofuran
T=20°C; 3 h;
2: p-toluenesulphonyl cyanide in tetrahydrofuran
参考文献
Poisson, Thomas; Oudeyer, Sylvain; Levacher, Vincent
Tetrahedron Letters, 2012 , vol. 53, # 26 p. 3284 - 3287