反应条件
1: N-(2-chloro-4-pyrimidinyl)-N-(3-methyl-1H-indazol-6-yl)amine With sodium hydride in N,N-dimethyl-formamide T=20°C; 0.25 h; 2: methyl iodide in N,N-dimethyl-formamide T=20°C; 0.5 h;
参考文献
Journal of Medicinal Chemistry, , vol. 51, # 15 p. 4632 - 4640