反应条件
1: 2,2,6,6-tetramethylpiperidinyl-lithium; iodine / tetrahydrofuran / -78 - 20 °C 2: sulfuric acid / 1,4-dioxane / 115 °C View Scheme
参考文献
Eastwood, Paul; Gonzalez, Jacob; Gomez, Elena; Caturla, Francisco; Aguilar, Nuria; Mir, Marta; Aiguade, Josep; Matassa, Victor; Balague, Cristina; Orellana, Adelina; Dominguez, Maria
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 21 p. 6253 - 6257