反应条件
1.1: 76 percent / EDCI; DMAP / CH2Cl2 / 2 h / 0 - 20 °C 2.1: Cl2Ru(PCy3)=(CHPh)(N,N'-Mes2-imidazolidin-2-yl) / CH2Cl2 / 5 h / 35 °C 2.2: 56 percent / nanosize Zn; AcOH / tetrahydrofuran / 0.17 h 3.1: 90 percent / HF*Py / tetrahydrofuran / 3 h / 20 °C 4.1: 86 percent / potassium diazodicarboxylate; AcOH / CH2Cl2 / Heating View Scheme
参考文献
Biswas, Kaustav; Lin, Hong; Njardarson, Jon T.; Chappell, Mark D.; Chou, Ting-Chao; Guan, Yongbiao; Tong, William P.; He, Lifeng; Horwitz, Susan B.; Danishefsky, Samuel J.
Journal of the American Chemical Society, 2002 , vol. 124, # 33 p. 9825 - 9832
