1: With 3-chloro-benzenecarboperoxoic acid in dichloromethane 42 h; Heating / reflux; 2: With sodium hydroxide; water 4 h; Heating / reflux; 3: With hydrogenchloride; water
参考文献
ASTEX THERAPEUTICS LIMITED; THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL; ASTRAZENECA AB
Patent: WO2006/136829 A2, 2006 ;
Location in patent: Page/Page column 123-124 ;
WO 2006/136829 A2