反应条件
1: 43 percent / CF3CO2H / CH2Cl2 / 4 h / 20 °C 2: 99 percent / (R)-tetrahydro-1-Me-3,3-Ph2-1H,3H-pyrrolo[1,2-c][1,3-2]oxaza; borole; BH3*THF / toluene / 5 - 20 °C 3: 70 percent / NaH / dimethylformamide / 3 h / 20 °C View Scheme
参考文献
Coe, Diane M; Perciaccante, Rossana; Procopiou, Panayiotis A
Organic and biomolecular chemistry, 2003 , vol. 1, # 7 p. 1106 - 1111