1-(2,3-二氢-3,3-二甲基-6-硝基-1H-吲哚-1-基)-乙酮合成路线 （共 12 条）
反应条件
1: NaH / dimethylformamide / 20 °C
2: 92 percent / HCOONa; Et4NCl*H2O; NaOAc / Pd(OAc)2 / dimethylformamide / 85 - 95 °C
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参考文献
Liu, Pingli; Huang, Liang; Lu, Yuelie; Dilmeghani, Mina; Baum, Jean; Xiang, Tingjian; Adams, Jeff; Tasker, Andrew; Larsen, Rob; Faul, Margaret M.
Tetrahedron Letters, 2007 , vol. 48, # 13 p. 2307 - 2310
反应条件
1: acetic anhydride / acetic acid
2: potassium carbonate / N,N-dimethyl-formamide
3: sodium formate; sodium acetate / palladium diacetate / N,N-dimethyl-formamide
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参考文献
Vertex Pharmaceuticals Incorported
Patent: US2011/98311 A1, 2011 ;
