反应条件
1: 1,8-diazabicyclo[5.4.0]undec-7-ene / acetonitrile / 2 h / 0 - 20 °C 2: potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride / N,N-dimethyl-formamide / 15 h / 85 °C View Scheme
参考文献
HANMI PHARMACEUTICAL CO., LTD.; Park, Chul Hyun; Kim, Won Jeoung; Jung, Young Hee; Kim, Nam Du; Chang, Young Kil; Kim, Maeng Sup
Patent: US2014/163226 A1, 2014 ;