反应条件
1: With sodium hydride in N,N-dimethyl-formamide; mineral oil T=-10°C; 3 h; Inert atmosphere; 2: With hydrogenchloride in water; N,N-dimethyl-formamide; mineral oil
参考文献
Yoshikawa, Kenji; Yokomizo, Aki; Naito, Hiroyuki; Haginoya, Noriyasu; Kobayashi, Shozo; Yoshino, Toshiharu; Nagata, Tsutomu; Mochizuki, Akiyoshi; Osanai, Ken; Watanabe, Kengo; Kanno, Hideyuki; Ohta, Toshiharu
Bioorganic and Medicinal Chemistry, 2009 , vol. 17, # 24 p. 8206 - 8220