3-氟溴苄合成路线

202197-31-75-氨基-1-(3-氟苄基)吲唑

参考文献

WO2011/2523 A1, ;
WO 2011/002523 A1

参考文献

Petrov, Kimberly G.; Zhang, Yue-Mei; Carter, Malcolm; Cockerill, G. Stuart; Dickerson, Scott; Gauthier, Cassandra A.; Guo, Yu; Mook Jr., Robert A.; Rusnak, David W.; Walker, Ann L.; Wood, Edgar R.; Lackey, Karen E.
Bioorganic and Medicinal Chemistry Letters, 2006 , vol. 16, # 17 p. 4686 - 4691

1155360-98-7+

456-41-73-氟溴苄

1155361-01-5

参考文献

Chai, Xiaoyun; Zhang, Jun; Hu, Honggang; Yu, Shichong; Sun, Qingyan; Dan, Zhigang; Jiang, Yuanying; Wu, Qiuye
European Journal of Medicinal Chemistry, 2009 , vol. 44, # 5 p. 1913 - 1920

参考文献

Jolidon, Synese; Rodriguez Sarmiento, Rosa Maria; Thomas, Andrew William; Wostl, Wolfgang; Wyler, Rene
Patent: US2004/34096 A1, 2004 ;

456-41-73-氟溴苄

70090-82-3

参考文献

Rafizadeh, Karim; Yates, Keith
Journal of Organic Chemistry, 1984 , vol. 49, # 9 p. 1500 - 1506

124-40-3二甲胺+

456-41-73-氟溴苄

770-18-3

参考文献

Liu, Zhongfa; Sayre, Lawrence M.
Tetrahedron, 2004 , vol. 60, # 7 p. 1601 - 1610

456-41-73-氟溴苄+

122-52-1亚磷酸三乙酯

80395-16-0

参考文献

Kawasaki, Takayasu; Saito, Koji; Ohta, Hiromichi
Chemistry Letters, 1997 , # 4 p. 351 - 352

456-41-73-氟溴苄+

5401-94-55-硝基吲唑

529508-58-51-[(3-氟苯基)甲基]-5-硝基-1H-吲唑+

833474-48-9

参考文献

BAYER PHARMACEUTICALS CORPORATION; ZHANG, Chengzhi
Patent: WO2006/23843 A2, 2006 ;
Location in patent: Page/Page column 104-105 ;

456-41-73-氟溴苄+

60-24-22-巯基乙醇

85582-62-32-[(3-氟苄基)硫基]乙醇

参考文献

UNIVERSITY OF STRATHCLYDE; UNIVERSITY OF GLASGOW; HARNETT, Margaret; HARNETT, William; SUCKLING, Professor Colin J; SCOTT, Fraser; HUGGAN, Judith Kerr; KHALAF, Abedawn Ibrahim
Patent: WO2014/23934 A1, 2014 ;
Location in patent: Page/Page column 18-19 ;

456-41-73-氟溴苄

865611-14-9

参考文献

De Candia, Modesto; Fiorella, Filomena; Lopopolo, Gianfranco; Carotti, Andrea; Romano, Maria Rosaria; Lograno, Marcello Diego; Martel, Sophie; Carrupt, Pierre-Alain; Belviso, Benny D.; Caliandro, Rocco; Altomare, Cosimo
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