反应条件
1: N,N-dimethylethylenediamine; potassium hydrophosphate; copper(l) iodide / toluene / 16 h / 25 - 80 °C 2: hydrogenchloride / 1,4-dioxane; dichloromethane / 3 h / 0 - 25 °C View Scheme
参考文献
LUPIN LIMITED; JANA, Gourhari; KURHADE, Sanjay, Pralhad; JAGDALE, Arun, Rangnath; KUKREJA, Gagan; SINHA, Neelima; PALLE, Venkata, P.; KAMBOJ, Rajender, Kumar
Patent: WO2014/9872 A1, 2014 ;