5-氟-2-(4,4,5,5-四甲基-1,3,2-二氧硼烷)-苯甲腈合成路线 (共 3 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane; dimethyl sulfoxide T=90°C; 18 h;
参考文献
WO2003/99816 A1, ;
Page 68-69 ;
WO 03/099816 A1
参考文献
US2004/132767 A1, ;
Page 12 ;
US 20040132767 A1
反应条件
potassium phosphate; tetrakis(triphenylphosphine) palladium(0) in N,N-dimethyl acetamide
T=65°C; 18 h;
参考文献
MERCK SHARP and DOHME LIMITED
Patent: WO2004/76452 A1, 2004 ;
Location in patent: Page 48 ;