1-异氰基-4-(三氟甲氧基)苯合成路线 (共 1 条)
反应条件
1.1: tetrahydrofuran / 60 °C
2.1: potassium tert-butylate / tert-butyl alcohol / 0.08 h / 30 °C
2.2: 1.5 h / 30 °C
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参考文献
CONVERGENCE PHARMACEUTICALS LIMITED; BESWICK, Paul John; GLEAVE, Robert James; HACHISU, Shuji; VILE, Sadie; BERTHELEME, Nicolas; WARD, Simon E
Patent: WO2012/4604 A1, 2012 ;
WO 2012/004604 A1