反应条件
1.1: AlCl3, aluminium chloride / chlorobenzene / Reflux 1.2: Cooling with ice 2.1: triphenylphosphine; di-tert-butylazodicarboxylate / tetrahydrofuran / 80 °C 3.1: AlCl3, aluminium chloride / dichloromethane / 0 - 10 °C 4.1: sodium hydroxide / tetrahydrofuran / 3 h / 20 °C View Scheme
参考文献
MAPI PHARMA HOLDINGS (CYPRUS) LIMITED; MAROM, Ehud; MIZHIRITSKII, Michael; RUBNOV, Shai
Patent: WO2011/99010 A1, 2011 ;
