反应条件
1: 81.2 percent / toluene / 1.) 5 h, RT; 2.) 4 d, RT
2: H2O / 1 h / 93 °C
3: 1.) 36percent HCl; 2.) NaOH / 1.) H2O, 2 h, RT; 2.) H2O, 10 deg C to 15 deg C
View Scheme
参考文献
Banholzer; Pook
Arzneimittel-Forschung/Drug Research, 1985 , vol. 35, # 1 A p. 217 - 228