反应条件
1: With 2,2,6,6-tetramethyl-piperidine; n-butyllithium in tetrahydrofuran T=-40°C; Inert atmosphere; 2: With hydrogenchloride; water T=80°C;
参考文献
Haga, Yuji; Sakamoto, Toshihiro; Shibata, Takunobu; Nonoshita, Katsumasa; Ishikawa, Makoto; Suga, Takuya; Takahashi, Hirobumi; Takahashi, Toshiyuki; Takahashi, Hidekazu; Ando, Makoto; Murai, Takashi; Gomori, Akira; Oda, Zenjun; Kitazawa, Hidefumi; Mitobe, Yuko; Kanesaka, Maki; Ohe, Tomoyuki; Iwaasa, Hisashi; Ishii, Yasuyuki; Ishihara, Akane; Kanatani, Akio; Fukami, Takehiro
Bioorganic and Medicinal Chemistry, 2009 , vol. 17, # 19 p. 6971 - 6982