1: With n-butyllithium in tetrahydrofuran; hexane
T=-78°C; 1 h;
2: With boric acid trimethyl ester in tetrahydrofuran; hexane
T=-78 - 20°C; 3.5 h;
3: With hydrogenchloride in tetrahydrofuran; hexane; water
参考文献
LG CHEM. LTD.
Patent: WO2007/69847 A1, 2007 ;
Location in patent: Page/Page column 29 ;