反应条件
1: With 2,2,6,6-tetramethyl-piperidine; n-butyllithium in tetrahydrofuran T=-78°C; 1 h; 2: With boric acid trimethyl ester in tetrahydrofuran T=-78°C; 2 h;
参考文献
MERCK SHARP and DOHME CORP.; ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.R.L.; MCCAULEY, John, A.; LIVERTON, Nigel, J.; RUDD, Michael, T.; GILBERT, Kevin, F.; FERRARA, Marco; SUMMA, Vincenzo; CRESCENZI, Benedetta
Patent: WO2012/40040 A1, 2012 ;
Location in patent: Page/Page column 45 ;
WO 2012/040040 A1