1-(5-氨基-2-吡啶)-4-羟基哌啶合成路线 (共 1 条)
反应条件
hydrogen; palladium 10 on activated carbon in ethanol
T=20°C; 3 h;
参考文献
BRISTOL-MYERS SQUIBB COMPANY; DEVASTHALE, Pratik; WASHBURN, William N.; RENDUCHINTALA, Kishore V.; SRIDHAR, Radhakrishnan
Patent: WO2010/42682 A1, 2010 ;
Location in patent: Page/Page column 71 ;
WO 2010/042682 A1