2-氯-2,2-二氟-1-(1H-吲哚-3-基)乙酮合成路线 (共 1 条)
反应条件
1: indole With diethylaluminium chloride in dichloromethane; toluene
T=0°C; 0.5 h;
2: difluorochloroacetyl chloride in dichloromethane; toluene
T=0°C; 2.5 h;
参考文献
Novartis AG
Patent: EP1783114 A1, 2007 ;
Location in patent: Page/Page column 24 ;