1: 71 percent / acetic anhydride / 0.5 h / 100 °C 2: conc. aq. HCl / 25 °C View Scheme
参考文献
Hoyte, Robert M.; Zhang, Jing-xin; Lerum, Ronald; Oluyemi, Aladejebi; Persaud, Prita; O'Connor, Craig; Labaree, David C.; Hochberg, Richard B.
Journal of Medicinal Chemistry, 2002 , vol. 45, # 24 p. 5397 - 5405