1-[4-溴-2-(羟基甲基)苯基]-4-(二甲基氨基)-1-(4-氟苯基)-1-丁醇盐酸盐(1:1)合成路线 (共 1 条)
反应条件
methanesulfonyl chloride; triethylamine in dichloromethane
T=-5 - 20°C; 2 - 3 h;
参考文献
Zhang, Peng; Cyriac, George; Kopajtic, Theresa; Zhao, Yongfang; Javitch, Jonathan A.; Katz, Jonathan L.; Newman, Amy Hauck
Journal of Medicinal Chemistry, 2010 , vol. 53, # 16 p. 6112 - 6121