5-氟-2-(甲氧基甲氧基)苯硼酸合成路线 (共 1 条)
反应条件
1: 2-bromo-4-fluoro-1-(methoxymethoxy)benzene With n-butyllithium in tetrahydrofuran; hexane T=-78°C; 1 h; 2: boric acid trimethyl ester in tetrahydrofuran; hexane T=-78 - 20°C; 2 h;
参考文献
WO2004/50637 A2, ;
Page 65-66 ;
WO 2004/050637 A2