反应条件
1: With anhydrous lithium acetate in N,N-dimethyl-formamide
T=20°C; 16 h;
2: With hydrogenchloride in N,N-dimethyl-formamide
T=-45°C;
3: With sodium tetrahydroborate; sodium hydrogencarbonate in methanol; N,N-dimethyl-formamide
T=-45 - 20°C;
参考文献
Kawano, Yoshikazu; Fujisawa, Hidehiko; Mukaiyama, Teruaki
Chemistry Letters, 2005 , vol. 34, # 4 p. 614 - 615