(4-氨基-3-氟-苯基)硼酸盐酸盐合成路线 （共 2 条）
反应条件
1.1: 47 percent / n-BuLi / tetrahydrofuran; hexane / 0 - 20 °C 2.1: t-BuLi / diethyl ether; pentane / -78 °C 2.2: trimethylborate / diethyl ether; tetrahydrofuran; pentane / -78 °C 2.3: 45 percent / HCl / diethyl ether; tetrahydrofuran; pentane / 20 °C View Scheme
参考文献
GENELABS TECHNOLOGIES, INC.
Patent: WO2006/76529 A1, 2006 ;
Location in patent: Page/Page column 161; 162 ;
反应条件
1: With potassium acetate; bis-triphenylphosphine-palladium(II) chloride in dimethyl sulfoxide T=60°C; 2: With water in dimethyl sulfoxide
参考文献
GENELABS TECHNOLOGIES, INC.
Patent: WO2008/8912 A1, 2008 ;
Location in patent: Page/Page column 97 ;
