7-氯-5-(2-氟苯基)-1,3-二氢-1-(2,2,2-三氟乙基)-2H-1,4-苯并二氮杂卓-2-酮合成路线 (共 2 条)
反应条件
Hg(CH3COO)2
T=20°C; 0.25 h; pH 11.2 (Britton-Robinson buffer); 40percent DMF as solubilisator;
参考文献
Oelschlaeger; Volke; Linde; Fedai; Schmidt
Archiv der Pharmazie, 1988 , vol. 321, # 8 p. 457 - 462
反应条件
sulfuric acid in acetonitrile
T=100°C; 2 h;
参考文献
Yang
Journal of Pharmaceutical Sciences, 1994 , vol. 83, # 1 p. 58 - 63