1: With sodium hydrogencarbonate in N,N-dimethyl-formamide
T=60°C; 16 h;
2: With hydrogenchloride in water; ethyl acetate; N,N-dimethyl-formamide
T=20°C; pH=3;
参考文献
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA; NATIONAL INSTITUTES OF HEALTH; COHEN, Seth M.; AGRAWAL, Arpita; DESOTO, Jamie; POMMIER, Yves; MADDALI, Kasthuraiah
Patent: WO2012/106534 A2, 2012 ;
Location in patent: Page/Page column 70 ;
WO 2012/106534 A2
Labbe, Genevieve; Krismanich, Anthony P.; De Groot, Sarah; Rasmusson, Timothy; Shang, Muhong; Brown, Matthew D.R.; Dmitrienko, Gary I.; Guillemette, J. Guy
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