反应条件
1: 88 percent / 25percent aq. NH3 / 6 h / 126 - 129 °C / 3800 - 9120 Torr 2: 3 h / 110 - 120 °C 3: 78.4 percent / 25percent aq. NH3 / 1.) 0-5 deg C, 2) 48-50 deg C, 10 h 4: dimethylaniline, POCl3 / toluene / 6 h / 83 - 87 °C View Scheme
参考文献
Yakhontov, L. N.; Zhikhareva, G. P.; Mastafanova, L. I.; Evstratova, M. I.; Pershin, G. N.; et al.
Pharmaceutical Chemistry Journal, 1987 , vol. 21, # 1 p. 34 - 45
Khimiko-Farmatsevticheskii Zhurnal, 1987 , vol. 21, # 1 p. 38 - 49