1: H2 / 10percent Pd/C / tetrahydrofuran / 3.5 h / 258.6 Torr / Ambient temperature
2: benzene; tetrahydrofuran / 8 h / Heating
View Scheme
参考文献
Collins, Paul W.; Gasiecki, Alan F.; Perkins, Willam E.; Gullikson, Gary W.; Jones, Peter H.; Bauer, Raymond F.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 5 p. 1001 - 1006