反应条件
1: 3-Fluoro-4-chlorophenol With potassium carbonate in N,N-dimethyl-formamide T=20°C; 0.25 h; 2: methyl iodide in N,N-dimethyl-formamide T=20°C;
参考文献
NEWLINK GENETICS; MAUTINO, Mario, R.; KUMAR, Sanjeev; JAIPURI, Firoz; WALDO, Jesse; KESHARWANI, Tanay; ZHANG, Xiaoxia
Patent: WO2011/56652 A1, 2011 ;
Location in patent: Page/Page column 118-119 ;
WO 2011/056652 A1