反应条件
1: 80 percent / p-TsOH, Et3O / dimethylformamide / Heating 2: 1.) aluminium trichloride; 2.) chlorotrimethylsilane / 1.) 1,2-dichloroethane, room temp., 1.5 h; 2.) 1,2-dichloroethane, room temp., 24 h, 80 deg C 28 h View Scheme
参考文献
Naora, Hirokazu; Ohnuki, Takashi; Nakamura, Asao
Bulletin of the Chemical Society of Japan, 1988 , vol. 61, # 7 p. 2401 - 2404