反应条件
1: 68 percent / triethylamine / acetonitrile / 0.5 h / Ambient temperature 2: 94 percent / triethylamine, p-toluenesulfonic acid, 4 Angstroem molecular sieves / acetonitrile / 16 h / Heating View Scheme
参考文献
Huang, Horng-Chih; Li, James J.; Garland, Danny J.; Chamberlain, Timothy S.; Reinhard, Emily J.; Manning, Robert E.; Seibert, Karen; Koboldt, Carol M.; Gregory, Susan A.; Anderson, Gary D.; Veenhuizen, Amy W.; Zhang, Yan; Perkins, William E.; Burton, Earl G.; Cogburn, J. Nita; Isakson, Peter C.; Reitz, David B.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 1 p. 253 - 266