反应条件
1: 2-(4-nitrophenyl)acetic acid With 1,1'-carbonyldiimidazole in dichloromethane
1 h;
2: toluene-4-sulfonamide in dichloromethane
1 h;
3: With 1,8-diazabicyclo[5.4.0]undec-7-ene in dichloromethane
16 h; Further stages.;
参考文献
Uehling, David E.; Donaldson, Kelly H.; Deaton, David N.; Hyman, Clifton E.; Sugg, Elizabeth E.; Barrett, David G.; Hughes, Robert G.; Reitter, Barbara; Adkison, Kim K.; Lancaster, Mary E.; Lee, Frank; Hart, Robert; Paulik, Mark A.; Sherman, Bryan W.; True, Timothy; Cowan, Conrad
Journal of Medicinal Chemistry, 2002 , vol. 45, # 3 p. 567 - 583
