2-氯-3-氟-[1,1-联苯]-4-羧酸合成路线 (共 1 条)
反应条件
potassium phosphate; tris-(dibenzylideneacetone)dipalladium(0); tri-cyclo-hexyl-phosphine in 1,4-dioxane
T=100°C; 1 h; Microwave irradiation;
参考文献
Choi, Jun Yong; Calvet, Claudia M.; Gunatilleke, Shamila S.; Ruiz, Claudia; Cameron, Michael D.; McKerrow, James H.; Podust, Larissa M.; Roush, William R.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 19 p. 7651 - 7668