反应条件
1: 2-amino-3-methoxy-benzoic acid With 1,1'-carbonyldiimidazole in N,N-dimethyl-formamide
T=40°C;
2: methylamine in N,N-dimethyl-formamide
T=20°C;
参考文献
Mizutani, Takashi; Nagase, Tsuyoshi; Ito, Sayaka; Miyamoto, Yasuhisa; Tanaka, Takeshi; Takenaga, Norihiro; Tokita, Shigeru; Sato, Nagaaki
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 23 p. 6041 - 6045