1: With sodium hydroxide in methanol
T=20°C; 0.5 h;
2: With hydrogenchloride in water
pH=3;
参考文献
CEPHALON, INC.; BRESLIN, Henry J.; CURRY, Matthew A.; GINGRICH, Diane E.; LEARN, Keith S.; OTT, Gregory R.; WAGNER, Jason C.
Patent: WO2013/116291 A1, 2013 ;
Location in patent: Page/Page column 225 ;