2-氯-N-甲基-5-(三氟甲基)嘧啶-4-胺合成路线 (共 1 条)
反应条件
triethylamine in methanol
T=-10 - 20°C;
参考文献
F. HOFFMANN-LA ROCHE AG; BAKER-GLENN, Charles; BURDICK, Daniel Jon; CHAMBERS, Mark; CHEN, Huifen; ESTRADA, Anthony; SWEENEY, Zachary Kevin; CHAN, Bryan K.
Patent: WO2012/62783 A1, 2012 ;
Location in patent: Page/Page column 68 ;
WO 2012/062783 A1