2,2-二甲基-2'-[(甲基氨基)硫代甲酰]丙酰肼合成路线 (共 2 条)
反应条件
methanesulfonic acid
1) 15 min, 25 deg C 2) reflux 4 h;
参考文献
Kress, Thomas J.; Costantino, Silvio M.
Journal of Heterocyclic Chemistry, 1980 , vol. 17, p. 607 - 608
反应条件
pyridine in tetrahydrofuran
T=20°C; 5 h; Reflux;
参考文献
Faridoon; Hussein, Waleed M.; Vella, Peter; Islam, Nazar Ul; Ollis, David L.; Schenk, Gerhard; McGeary, Ross P.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 1 p. 380 - 386