反应条件
1: 85 percent / AlCl3 / 1,2-dichloro-ethane / 1) 0-5 deg C -> r.t., 2 h 2) reflux, 1h
2: NH2OH*HCl, pyridine / 4 h / Heating
View Scheme
参考文献
Sato; Dan; Onuma; Tanaka; Aoki; Koga
Chemical and Pharmaceutical Bulletin, 1991 , vol. 39, # 7 p. 1760 - 1772