4-氟-3-碘-1H-吲唑合成路线 (共 1 条)
反应条件
iodine; potassium hydroxide in N,N-dimethyl-formamide T=20°C; 2 h;
参考文献
MERCK SHARP and DOHME CORP.; BARR, Kenneth Jay; MACLEAN, John; ZHANG, Hongjun; BERESIS, Richard Thomas; ZHANG, Dongshan
Patent: WO2014/28597 A2, 2014 ;
Location in patent: Page/Page column 59 ;