反应条件
1: 1.) NaH / 1.) DMF, 0 deg C, 1 h, 2.) DMF, 0 deg C, 3 h
2: dimethylformamide / 2 h / 0 - 20 °C
3: HCl / dioxane
View Scheme
参考文献
Rosenberg; Spina; Woods; Polakowski; Martin; Yao; Stein; Cohen; Barlow; Egan; Tricarico; Baker; Kleinert
Journal of Medicinal Chemistry, 1993 , vol. 36, # 4 p. 449 - 459