反应条件
1: hydrogenchloride / 1,2-dichloro-benzene / 12 h / 20 °C
2: potassium carbonate / N,N-dimethyl-formamide / 6 h / 20 °C
3: sodium hydroxide / tetrahydrofuran; water / 3 h / 20 °C
4: 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride / dichloromethane / 3 h / 20 °C
View Scheme
参考文献
Gathirwa, Jeremiah W.; Maki, Toshihide
Synthetic Communications, 2013 , vol. 43, # 7 p. 1016 - 1022