反应条件
1: palladium diacetate; triethylamine; tris-(o-tolyl)phosphine / N,N-dimethyl-formamide / 4 h / 120 °C
2: palladium diacetate; potassium formiate / N,N-dimethyl-formamide / 29 h
3: trifluoroacetic acid / dichloromethane / 1 h / 20 °C
View Scheme
参考文献
Matsuo, Kazuya; Nakagawa, Hidehiko; Adachi, Yusuke; Kameda, Eri; Aizawa, Kazuyuki; Tsumoto, Hiroki; Suzuki, Takayoshi; Miyata, Naoki
Chemical and Pharmaceutical Bulletin, 2012 , vol. 60, # 8 p. 1055 - 1062