7-溴吡啶并[2,3-b]吡嗪合成路线

参考文献

WO2010/52448 A2, ;

Page/Page column 41-42 ;
WO 2010/052448 A2

52333-42-37-溴吡啶并[2,3-b]吡嗪

322-46-32,3-二吡啶吡嗪

参考文献

Leese; Rydon
Journal of the Chemical Society, 1955 , p. 303,307

52333-42-37-溴吡啶并[2,3-b]吡嗪+

73183-34-3联硼酸频那醇酯

1210047-44-1吡啶并[2,3-b]吡嗪-7-基硼酸频那醇酯

参考文献

BAYER SCHERING PHARMA AKTIENGESELLSCHAFT; BAeRFACKER, Lars; KAST, Raimund; GRIEBENOW, Nils; MEIER, Heinrich; KOLKHOF, Peter; ALBRECHT-KUePPER, Barbara; NITSCHE, Adam; STASCH, Johannes-Peter; SCHNEIDER, Dirk; TEUSCH, Nicole; RUDOLPH, Joachim; WHELAN, James; BULLOCK, William; PLEASIC-WILLIAMS, Susan
Patent: WO2010/20363 A1, 2010 ;
Location in patent: Page/Page column 67-68 ;

52333-42-37-溴吡啶并[2,3-b]吡嗪

397325-35-8(9CI)-7-甲基吡啶并[2,3-b]吡嗪

参考文献

Sumitomo Pharmaceuticals Company, Limited
Patent: EP1479384 A1, 2004 ;

52333-42-37-溴吡啶并[2,3-b]吡嗪+

4542-61-4硼酸二甲酯+

144-55-8碳酸氢钠+

32005-36-0双(二亚芐基丙酮)钯

397325-35-8(9CI)-7-甲基吡啶并[2,3-b]吡嗪

参考文献

Tokunaga, Teruhisa; Hume, William Ewan; Kitoh, Makoto; Nagata, Ryu
Patent: US2003/181496 A1, 2003 ;