反应条件
<b>Multi-step reaction with 2 steps<br /> </b>1: K<sub>2</sub>CO<sub>3</sub> / dimethylformamide / 5 h / 40 - 50 °C<br />2: NaBH<sub>4</sub>, 0.5N aq.NaOH / tetrahydrofuran / 2.5 h / Ambient temperature<br /> <br />
参考文献
Nakazato, Atsuro; Ohta, Kohmei; Sekiguchi, Yoshinori; Okuyama, Shigeru; Chaki, Shigeyuki; Kawashima, Yutaka; Hatayama, Katsuo Journal of Medicinal Chemistry, 1999 , vol. 42, # 6 p. 1076 - 1087