反应条件
1: butan-1-ol / 4 h / 110 °C 2: 1 N HCl / 3 h / 50 °C 3: 52.5 percent / NaBH3CN, HCl, 3 Angstroem molecular sieves / methanol / 24 h / Ambient temperature View Scheme
参考文献
Dhainaut, Alain; Regnier, Gilbert; Atassi, Ghanem; Pierre, Alain; Leonce, Stephane; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 13 p. 2481 - 2496