反应条件
1: 1.) Piv-Cl, pyridine 2.) citric acid / 1.) THF, -15 - 0 deg C, 1 h 5 min 2.) water 2: H2 / Pd/C / tetrahydrofuran; acetic acid View Scheme
参考文献
Anteunis, M.J.O.; Becu, Chr.; Becu, F.
Bulletin des Societes Chimiques Belges, 1987 , vol. 96, # 2 p. 133 - 136