5-[(3-甲基苯基)氨基]-1,3,4-噻二唑-2(3H)-硫酮合成路线 （共 3 条）
反应条件
1: 1.) Mg / 1.) THF, reflux, 1 h, 2.) THF, RT, 2 h
2: PCl5 / CH2Cl2 / 1 h / Ambient temperature
3: ethanol / 1 h / Ambient temperature
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参考文献
Hogberg; Ulff; Renyi; Ross
Journal of Medicinal Chemistry, 1981 , vol. 24, # 12 p. 1499 - 1507
反应条件
sodium hydroxide; aluminium trichloride in o-di-fluorobenzene; di-isopropyl ether; pentane
参考文献
Laboratories UPSA
Patent: US5807873 A1, 1998 ;
反应条件
aluminium trichloride
T=85°C; 2 h;
参考文献
Langhals, Elke; Langhals, Heinz; Ruechardt, Christoph
Liebigs Annalen der Chemie, 1982 , # 5 p. 930 - 949
