反应条件
1: POCl3, PCl5 / toluene / 3.5 h / 95 - 110 °C
2: H2, glacial acetic acid / 10percent Pd/C / 0.5 h / 3000.2 Torr
View Scheme
参考文献
Santangelo; Casagrande; Miragoli; Vecchietti
European Journal of Medicinal Chemistry, 1994 , vol. 29, # 11 p. 877 - 882