反应条件
1: With sodium tris(acetoxy)borohydride; acetic acid in 1,2-dichloro-ethane
T=20°C;
2: With sodium hydrogencarbonate in water; 1,2-dichloro-ethane
参考文献
MITSUBISHI TANABE PHARMA CORPORATION; SANOFI-AVENTIS; WATANABE, Kazutoshi; NAKAYAMA, Kazuki; SAKAI, Daiki
Patent: WO2010/114179 A1, 2010 ;
Location in patent: Page/Page column 30 ;
WO 2010/114179 A1